2009
https://www.tandfonline.com/doi/full/10.3109/14756360903489581
Effects of some drugs on human erythrocyte glucose 6-phosphate dehydrogenase: an in vitro study
(2010). Effects of some drugs on human erythrocyte glucose 6-phosphate dehydrogenase: an in vitro study. Journal of Enzyme Inhibition and Medicinal Chemistry: Vol. 25, No. 6, pp. 871-875.
www.tandfonline.com
Effects of some drugs on human erythrocyte glucose 6-phosphate dehydrogenase: an in vitro study
Table II. IC50 values and Ki constants obtained from inhibition percent values vs five different inhibitors
Drugs IC50 (mM) Ki (mM) Inhibition type
| Ketotifen | 0.008 | 0.0052 ± 0.0012 | Non-competitive |
| Dacarbazine | 0.021 | 0.0154 ± 0.0011 | Non-competitive |
| Thiocolchicoside | 0.056 | 0.0397 ± 0.0063 | Non-competitive |
| Meloxicam | 0.067 | 0.0579 ± 0.0061 | Non-competitive |
| Methotrexat | 0.114 | 0.0910 ± 0.0166 | Non-competitive |
| Furosemide | 0.315 | 0.1874 ± 0.0136 | Non-competitive |
| Olanzapine | 0.53 | 0.4972 ± 0.0710 | Non-competitive |
| Methylprednizolone acetate | 2.23 | 0.5405 ± 0.1528 | Competitive |
| Paricalcitol | 2.28 | 4.2867 ± 1.0670 | Non-competitive |
| Ritodrine hydrochloride | 8.11 | 8.2081 ± 1.3522 | Non-competitive |
| Gadobenate-dimeglumine | 115 | 48.4380 ± 2.176 | Non-competitive |
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